SCHEMBL2420190

SCHEMBL2420190

COc1ccc(CSOSCc2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.61
ATM Q13315 2/20 0.53
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 3/20 0.52
PPARG P37231 1/20 0.52
PPARD Q03181 1/20 0.52
PPARA Q07869 1/20 0.52
POLB P06746 2/20 0.50
CYP19A1 P11511 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
AOC3 Q16853 1/20 0.47
LDHA P00338 1/20 0.47
SIGMAR1 Q99720 1/20 0.46
STAT3 P40763 1/20 0.46
MAPT P10636 3/20 0.45
GAA P10253 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2420183 0.83 CA2 (0.65) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL28509107 0.82 MEN1 (0.56) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL31157848 0.76 CYP19A1 (0.77) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL16641094 0.76 CYP19A1 (0.77) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL2095593 0.76 CA2 (1.00) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL11444350 0.76 CA2 (0.55) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL11192594 0.74 CA2 (0.53) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL31275634 0.74 CA2 (0.71) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL27442665 0.74 CA2 (0.71) CA2ATMKDM4EALDH1A1PPARG
SCHEMBL31428 0.74 CA2 (0.71) CA2ATMKDM4EALDH1A1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013083541-A1 (4-MERCAPTO-PIPERIDIN-4-YL)-AMINOACETIC ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF LACER, S.A. (ES) 2013-06-13 WO disclosed
EP-2601940-A1 (4-mercapto-piperidin-4-yl)-aminoacetic acid derivatives, pharmaceutical compositions and uses thereof LACER, S.A. (ES) 2013-06-12 EP disclosed
EP-2125727-B1 STABLE S-NITROSOTHIOLS, METHOD OF SYNTHESIS AND USE LACER SA (ES) 2012-11-21 EP disclosed
CN-101600692-B Stable s-nitrosothiols, method of synthesis and use LACER SA ES 2012-07-04 CN disclosed
US-8012993-B2 e.g. ethyl(R,S)-acetylamino-(1-methyl-4-S-nitrosomercapto-piperidin-4-yl)-acetate; vasodilating effect which inhibit the aggregation of the platelets; hypotensive agent, vasodilator; thrombosis, graft rejections, ischemia-reperfusion; adding mercaptan compound to heterocyclic followed by nitrosation LACER, S.A. (ES) 2011-09-06 US disclosed
CN-101600692-A Stable S-nitrosothiol, preparation method and use LACER SA (ES) 2009-12-09 CN disclosed
EP-2125727-A1 STABLE S-NITROSOTHIOLS, METHOD OF SYNTHESIS AND USE LACER, S.A. (ES) 2009-12-02 EP disclosed
WO-2008080986-A1 FURAN DERIVATIVES, METHOD OF SYNTHESIS AND USES THEREOF NEUROPHARMA, S.A. (ES) 2008-07-10 WO disclosed
WO-2008080934-A1 STABLE S-NITROSOTHIOLS, METHOD OF SYNTHESIS AND USE LÁCER, S.A. (ES) 2008-07-10 WO disclosed
US-20080161354-A1 STABLE S-NITROSOTHIOLS, METHOD OF SYNTHESIS AND USE LACER, S.A. (ES) 2008-07-03 US disclosed
EP-1939179-A1 Stable S-nitrosothiols, method of synthesis and use LACER, S.A. (ES) 2008-07-02 EP disclosed
EP-1939191-A1 Furan derivatives, method of synthesis and uses thereof Neuropharma S.A. (ES) 2008-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161354-A1 STABLE S-NITROSOTHIOLS, METHOD OF SYNTHESIS AND USE NOS2, PTGIS, NOS1 CA2 2151/4885ATM 2520/4885KDM4E 4245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.