SCHEMBL242048

SCHEMBL242048

O=C=Nc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 5/20 0.50
TSHR P16473 2/20 0.50
CYP3A4 P08684 1/20 0.47
NR1H2 P55055 1/20 0.45
BAX Q07812 1/20 0.45
MAOA P21397 1/20 0.45
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
GSTP1 P09211 1/20 0.42
SOS1 Q07889 1/20 0.42
CA9 Q16790 1/20 0.42
PARP10 Q53GL7 1/20 0.42
MIF P14174 1/20 0.41
SRD5A2 P31213 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
MGLL Q99685 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylether SCHEMBL28412262 0.92 LTA4H (0.46) LTA4HTSHRCYP3A4NR1H2BAX
SCHEMBL50333 0.91 CYP3A4 (0.54) LTA4HTSHRCYP3A4CA1CA2
SCHEMBL4544188 0.91 CYP3A4 (0.54) LTA4HTSHRCYP3A4CA1CA2
SCHEMBL4551613 0.91 CYP3A4 (0.54) LTA4HTSHRCYP3A4CA1CA2
SCHEMBL8700318 0.91 LTA4H (0.41) LTA4HTSHRCYP3A4NR1H2BAX
SCHEMBL7136291 0.88 FURIN (0.53) TSHRCYP3A4PARP10
Diphenylmethane SCHEMBL2583973 0.87 CYP3A4 (0.63) LTA4HTSHRCYP3A4SRD5A2
SCHEMBL28101747 0.87 PPARG (0.42) LTA4HTSHRCYP3A4MAOAMIF
SCHEMBL22966366 0.86 MAPT (0.43) LTA4HTSHRCYP3A4NR1H2BAX
SCHEMBL1415412 0.85 CYP3A4 (0.48) LTA4HTSHRCYP3A4GSTP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 620 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117926640-A Environment-friendly decorative paper and preparation method thereof 浙江锦尚添彩新材料有限公司 2024-04-26 CN claimed
CN-113354778-B Solid polycarboxylate superplasticizer and preparation method thereof 中建西部建设建材科学研究院有限公司 2023-10-03 CN claimed
CN-113354778-A Solid polycarboxylic acid water reducing agent and preparation method thereof 中建西部建设建材科学研究院有限公司 2021-09-07 CN claimed
EP-1761554-A2 PEPTIDE ANTIBIOTICS AND METHODS FOR MAKING SAME Biosource Pharm, Inc. (US) 2007-03-14 EP claimed
WO-2006083317-A2 PEPTIDE ANTIBIOTICS AND METHODS FOR MAKING SAME BIOSOURCE PHARM, INC. (US) 2006-08-10 WO claimed
EP-1377589-B1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS PHARMACIA ITALIA SPA (IT) 2005-09-07 EP claimed
EP-0215841-B1 PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION RHONE-POULENC NEDERLAND B.V. (NL) 1988-11-17 EP claimed
EP-0215841-A1 PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION. UNION CARBIDE CORP (US) 1987-04-01 EP claimed
EP-0215056-A1 PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION UNION CARBIDE CORPORATION (US) 1987-03-25 EP claimed
WO-1986005780-A1 PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION UNION CARBIDE CORPORATION (US) 1986-10-09 WO claimed
WO-1986005781-A1 PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION UNION CARBIDE CORPORATION (US) 1986-10-09 WO claimed
WO-2026104221-A1 PROCESS FOR PREPARING OF ORGANIC CARBAMOYL AZIDES All4Labels Group GmbH (DE) 2026-05-21 WO disclosed
EP-4713378-A1 ESTERIFIED ETHANOLAMINES FOR PREPARING ISOCYANURATE POLYMERS Covestro Deutschland AG (DE) 2026-03-25 EP disclosed
WO-2025104079-A1 SALICYLIC ACID AND PICOLINIC ACID DERIVATIVES AS INHIBITORS OF ENERGY COUPLING FACTOR (ECF) TRANSPORTERS FOR THE TREATMENT OF BACTERIAL INFECTIONS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2025-05-22 WO disclosed
CN-117926640-B Environment-friendly decorative paper and preparation method thereof 浙江锦尚添彩新材料有限公司 2025-05-06 CN disclosed
US-4033912-A Process for molding polyurethane foams BAYER AKTIENGESELLSCHAFT (DT) 1977-07-05 US disclosed
US-4005223-A Insecticidal 2-chloro-4'-[N-(N'-benzoyl)-ureido]-diphenyl ethers BAYER AKTIENGESELLSCHAFT (DT) 1977-01-25 US disclosed
US-4001256-A PROSTAGLANDIN PRODUCTION IN MAMMALS THE UPJOHN COMPANY (US) 1977-01-04 US disclosed
US-3992553-A Benzoylureido-diphenyl ether insecticides BAYER AKTIENGESELLSCHAFT (DT) 1976-11-16 US disclosed
US-3933814-A ANTIPROTOZOA, ANTICOCCIDIOSIS BAYER AKTIENGESELLSCHAFT (DT) 1976-01-20 US disclosed