SCHEMBL2421608

SCHEMBL2421608

CCOc1cc(C=O)c(-c2nccc3ccccc23)c(OCC)c1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.45
LMNA P02545 1/20 0.41
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 2/20 0.35
G6PD P11413 1/20 0.35
ALOX5 P09917 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SCN9A Q15858 1/20 0.34
S1PR3 Q99500 1/20 0.33
PTK6 Q13882 1/20 0.33
HTR2C P28335 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ERN1 O75460 1/20 0.33
SLC2A1 P11166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2417097 0.87 S1PR1 (0.43) S1PR1LMNAALDH1A1GAAMEN1
SCHEMBL2421361 0.80 MEN1 (0.42) S1PR1LMNAALDH1A1GAAMEN1
SCHEMBL2417802 0.80 GAA (0.42) S1PR1ALDH1A1GAAMEN1KMT2A
SCHEMBL2414362 0.79 GAA (0.41) S1PR1LMNAALDH1A1GAAMEN1
SCHEMBL2424612 0.74 GAA (0.41) S1PR1ALDH1A1GAAMEN1KMT2A
SCHEMBL2424610 0.74 L3MBTL1 (0.40) S1PR1ALDH1A1GAAMEN1KMT2A
Hydrochloric Acid SCHEMBL7343358 0.71 KMT2A (0.66) S1PR1LMNAALDH1A1GAAMEN1
SCHEMBL2417832 0.71 GAA (0.48) S1PR1LMNAALDH1A1GAAMEN1
SCHEMBL22946244 0.69 LMNA (0.58) LMNAALDH1A1GAAPOLBHPGD
SCHEMBL29633534 0.69 LMNA (0.58) LMNAALDH1A1GAAPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8026255-B2 Substituted piperidines as somatostatin receptor subtype 5 (SSTR5) antagonists HOFFMAN-LA ROCHE INC. (US) 2011-09-27 US disclosed