SCHEMBL24246191

SCHEMBL24246191

CCc1cccc2c1cc(Cc1cc(C)c3cc(C)n(C)c3c1C)n2C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
NQO2 P16083 1/20 0.35
NPEPPS P55786 1/20 0.34
ALKBH5 Q6P6C2 1/20 0.33
FTO Q9C0B1 1/20 0.33
CMA1 P23946 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
EGFR P00533 2/20 0.31
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22434745 0.78 NPEPPS (0.46) KDM4ENQO2NPEPPSALKBH5FTO
SCHEMBL20505366 0.64 KDM4E (0.41) KDM4ENPEPPSTSHRALDH1A1LMNA
SCHEMBL13548554 0.62 ALKBH5 (0.52) KDM4ENQO2ALKBH5FTOCYP1A2
SCHEMBL19557282 0.62 NPEPPS (0.42) KDM4ENQO2NPEPPSTSHRALDH1A1
SCHEMBL24246102 0.61 NOTUM (0.30)
SCHEMBL22434882 0.61 KCNH2 (0.33) MAPT
SCHEMBL23095471 0.60 NPEPPS (0.50) KDM4ENQO2NPEPPS
SCHEMBL11702583 0.60 ALKBH5 (0.59) KDM4ENQO2NPEPPSALKBH5FTO
SCHEMBL20759268 0.59 RAB9A (0.40) KDM4EALDH1A1LMNAMAPT
SCHEMBL25171221 0.59 DHFR (0.42) KDM4ENQO2NPEPPSALKBH5FTO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220175775-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2022-06-09 US disclosed
US-11241431-B2 N-substituted indole derivatives as PGE2 receptor modulators IDORSIA PHARMACEUTICALS LTD (CH) 2022-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220175775-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS PTGER1, PTGER4, PTGER2 KDM4E 2755/4885NQO2 693/4885NPEPPS 4104/4885
US-11241431-B2 N-substituted indole derivatives as PGE2 receptor modulators PTGER1, PTGER4, PTGER2 KDM4E 2755/4885NQO2 693/4885NPEPPS 4104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.