SCHEMBL24251664

SCHEMBL24251664

C=C(C)CNc1ccc(Cl)nc1C

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
GRM1 Q13255 2/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24496623 0.83 CCNA2 (0.32) CYP1A2CYP2C9TSHRCYP2C19GRM1
SCHEMBL24251705 0.83 CCNA2 (0.33) CYP1A2CYP2C9TSHRCYP2C19GRM1
SCHEMBL20680456 0.82 CCNA2 (0.34) CYP1A2CYP2C9TSHRCYP2C19GRM1
SCHEMBL29598023 0.82 CCNA2 (0.34) CYP1A2CYP2C9TSHRCYP2C19GRM1
SCHEMBL1642783 0.77 LMNA (0.38) TSHRALDH1A1KDM4EGAASMN1; SMN2
SCHEMBL24251663 0.76 LMNA (0.39) KDM4EGAA
SCHEMBL24496571 0.75 CYP1A2 (0.36) CYP1A2CYP2C9TSHRCYP2C19
SCHEMBL24251774 0.74 IAPP (0.43) CYP1A2CYP2C9TSHRCYP2C19CCNA2
SCHEMBL13947192 0.74 IDO1 (0.39) ALDH1A1KDM4EGAASMN1; SMN2MAPT
SCHEMBL13044666 0.72 ESR1 (0.44) TSHRALDH1A1KDM4EGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4257584-A1 2,3-DIHYDRO-1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Abbisko Therapeutics Co., Ltd. (CN) 2023-10-11 EP disclosed
WO-2023011505-A1 PYRIMIDINE OR PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN PHARMACY 上海和誉生物医药科技有限公司 2023-02-09 WO disclosed
WO-2022116995-A1 2,3-DIHYDRO-1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2022-06-09 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed