SCHEMBL24251705

SCHEMBL24251705

C=C(C)CNc1ccc(C)nc1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
GRM1 Q13255 1/20 0.31
LMNA P02545 2/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CCR1 P32246 1/20 0.30
RAB9A P51151 1/20 0.30
CCR5 P51681 1/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24496623 0.83 CCNA2 (0.32) CCNA2CDK2ALDH1A1CYP1A2CYP2C9
SCHEMBL24251715 0.83 CCNA2 (0.32) CCNA2CDK2ALDH1A1KDM4EGRM1
SCHEMBL24251664 0.83 CYP1A2 (0.37) CCNA2CDK2ALDH1A1KDM4ECYP1A2
SCHEMBL24251663 0.79 LMNA (0.39) KDM4ELMNAHTTKMT2ARAB9A
SCHEMBL24251774 0.77 IAPP (0.43) CCNA2CDK2ALDH1A1KDM4ECYP1A2
SCHEMBL24496546 0.74 P2RX7 (0.40) CCNA2CDK2ALDH1A1KDM4EGRM1
SCHEMBL13947026 0.72 IDO1 (0.41) ALDH1A1HTTCCR1RAB9ACCR5
SCHEMBL19122563 0.71 NPSR1 (0.51) ALDH1A1LMNAKMT2ASMN1; SMN2RAB9A
SCHEMBL24496571 0.71 CYP1A2 (0.36) CYP1A2CYP2C9TSHRCYP2C19
SCHEMBL13044656 0.70 IDO1 (0.42) ALDH1A1KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011505-A1 PYRIMIDINE OR PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN PHARMACY 上海和誉生物医药科技有限公司 2023-02-09 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed