SCHEMBL24251663

SCHEMBL24251663

C=C(C)CNc1ccc(C(F)(F)F)nc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
GAA P10253 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
KDM4E B2RXH2 2/20 0.33
CXCR4 P61073 1/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
PLK1 P53350 1/20 0.33
P2RX7 Q99572 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
KCNJ11 Q14654 1/20 0.32
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24996463 0.85 LMNA (0.34) LMNAPLK1P2RX7CA12CA1
SCHEMBL24251705 0.79 CCNA2 (0.33) LMNARAB9AKDM4EHTTKMT2A
SCHEMBL24251664 0.76 CYP1A2 (0.37) GAAKDM4E
SCHEMBL24496623 0.76 CCNA2 (0.32)
SCHEMBL8171101 0.73 LMNA (0.43) LMNANPC1RAB9AGAATRPV1
SCHEMBL10124516 0.73 LMNA (0.51) LMNANPC1RAB9AGAATRPV1
SCHEMBL24251774 0.71 IAPP (0.43) LMNANPC1RAB9AKDM4EMEN1
SCHEMBL25037178 0.69 LMNA (0.47) LMNANPC1RAB9AGAATRPV1
SCHEMBL25037262 0.69 ALDH1A1 (0.48) LMNANPC1RAB9AGAATRPV1
SCHEMBL25037266 0.69 LMNA (0.47) LMNANPC1RAB9AGAATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011505-A1 PYRIMIDINE OR PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN PHARMACY 上海和誉生物医药科技有限公司 2023-02-09 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed