SCHEMBL24251774

SCHEMBL24251774

C=C(C)CNc1ccc(C(=O)OC)nc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IAPP P10997 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.36
TP53 P04637 2/20 0.36
CYP1A2 P05177 2/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PTGER4 P35408 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TSHR P16473 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24251776 0.84 IAPP (0.45) IAPPSMN1; SMN2MAPTMAPK1TP53
SCHEMBL24251705 0.77 CCNA2 (0.33) SMN1; SMN2CYP1A2CYP2C9CYP2C19RAB9A
SCHEMBL24251664 0.74 CYP1A2 (0.37) SMN1; SMN2MAPTCYP1A2CYP2C9CYP2C19
SCHEMBL24496623 0.74 CCNA2 (0.32) CYP1A2CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL1161278 0.71 MAPT (0.48) SMN1; SMN2MAPTMAPK1TP53CYP1A2
SCHEMBL24251663 0.71 LMNA (0.39) NPC1RAB9AKDM4ELMNAHSD17B10
SCHEMBL9089861 0.70 MAPK1 (0.44) IAPPSMN1; SMN2MAPTMAPK1TP53
SCHEMBL23554282 0.70 MAPT (0.55) SMN1; SMN2MAPTMAPK1TP53CYP1A2
SCHEMBL16372000 0.70 LCK (0.47) SMN1; SMN2MAPTMAPK1TP53CYP1A2
SCHEMBL29549633 0.70 MAPT (0.55) SMN1; SMN2MAPTMAPK1TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed