SCHEMBL24253592

SCHEMBL24253592

O=C1CC(F)CC2(CCNCC2)N1c1ccc(Cl)c(F)c1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.33
RAD51 Q06609 1/20 0.33
SLC6A2 P23975 8/20 0.32
SLC6A4 P31645 8/20 0.32
SLC6A3 Q01959 8/20 0.32
MMP2 P08253 2/20 0.31
ADAMTS5 Q9UNA0 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4D Q08499 1/20 0.31
ADRB1 P08588 1/20 0.31
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24253912 0.89 BPTF (0.37) CYP11B2ADAMTS5
SCHEMBL24253590 0.87 MMP2 (0.33) CYP11B2RAD51SLC6A2SLC6A4SLC6A3
SCHEMBL26307735 0.86 MAPT (0.33) ADAMTS5PDE4BPDE4DADRB1
SCHEMBL24253513 0.80 SLC6A3 (0.36) CYP11B2RAD51SLC6A2SLC6A4SLC6A3
SCHEMBL30423624 0.80 SLC6A3 (0.36) CYP11B2RAD51SLC6A2SLC6A4SLC6A3
SCHEMBL30423977 0.76 TSHR (0.39) CYP11B2ADAMTS5
SCHEMBL24253711 0.76 TSHR (0.39) CYP11B2ADAMTS5
Hydrochloric Acid SCHEMBL30494641 0.75 TSHR (0.38) ADAMTS5
SCHEMBL26307724 0.74 RAD51 (0.39) CYP11B2RAD51SLC6A2SLC6A4SLC6A3
SCHEMBL26307736 0.74 CCR1 (0.33) ADAMTS5ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2022-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof REN, NR3C2, PKD1 CYP11B2 22/4885RAD51 3303/4885SLC6A2 851/4885
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF REN, NR3C2, PKD1 CYP11B2 22/4885RAD51 3303/4885SLC6A2 851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.