SCHEMBL30423977

SCHEMBL30423977

O=C1CC(O)CC2(CCNCC2)N1c1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
BPTF Q12830 1/20 0.36
HSD11B1 P28845 1/20 0.32
ADAMTS5 Q9UNA0 2/20 0.32
MMP13 P45452 1/20 0.32
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
ROCK2 O75116 1/20 0.31
POLB P06746 1/20 0.31
RAF1 P04049 1/20 0.31
BRAF P15056 1/20 0.31
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24253711 1.00 TSHR (0.39) TSHRBPTFHSD11B1ADAMTS5MMP13
Hydrochloric Acid SCHEMBL30494641 0.99 TSHR (0.38) TSHRBPTFHSD11B1ADAMTS5MMP13
SCHEMBL26307736 0.90 CCR1 (0.33) TSHRADAMTS5ROCK2
SCHEMBL24253590 0.90 MMP2 (0.33) ADAMTS5MMP13CYP11B2
SCHEMBL24253912 0.86 BPTF (0.37) TSHRBPTFADAMTS5MMP13HTR1A
SCHEMBL24253768 0.80 HSD11B1 (0.34) TSHRBPTFHSD11B1ADAMTS5MMP13
SCHEMBL30494563 0.77 ADAMTS5 (0.41) ADAMTS5MMP13ROCK2
SCHEMBL24253710 0.77 HTR1A (0.36) TSHRBPTFMMP13HTR1ADRD2
SCHEMBL24253592 0.76 CYP11B2 (0.33) ADAMTS5CYP11B2
SCHEMBL26307735 0.76 MAPT (0.33) ADAMTS5ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116157404-A Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof 诺华股份有限公司 2023-05-23 CN disclosed