SCHEMBL24253788

SCHEMBL24253788

CCc1cc(OC(=O)N2CCC(N3CCCCC3)CC2)ccc1Nc1cc(-c2ccc(-n3cccn3)cc2)n(C(=O)OC(C)(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.41
TNIK Q9UKE5 1/20 0.39
PIK3CD O00329 1/20 0.36
CYP2D6 P10635 2/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.35
CACNB4 O00305 1/20 0.35
CACNA1A O00555 1/20 0.35
CACNA1G O43497 1/20 0.35
CACNG3 O60359 1/20 0.35
CACNA1F O60840 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNB3 P54284 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CACNG7 P62955 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1D Q01668 1/20 0.35
CACNB1 Q02641 1/20 0.35
CACNG1 Q06432 1/20 0.35
CACNB2 Q08289 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24253982 0.83 TNIK (0.39) GPR119TNIKPIK3CD
SCHEMBL24253785 0.83 TNIK (0.60) TNIK
SCHEMBL24254069 0.77 TNIK (0.37) GPR119TNIKCYP2D6CYP1A2CYP3A4
SCHEMBL24253780 0.73 CYP2D6 (0.48) CYP2D6CYP1A2MAPTCYP3A4ALDH1A1
SCHEMBL24253879 0.70 TNIK (0.60) TNIK
SCHEMBL24254072 0.68 TNIK (0.56) TNIK
SCHEMBL24253816 0.67 GPR119 (0.46) GPR119PIK3CDMAPTJAK2JAK3
SCHEMBL24253971 0.65 CYP2D6 (0.48) CYP2D6CYP1A2MAPTCYP3A4ALDH1A1
SCHEMBL24253970 0.65 CYP2D6 (0.58) CYP2D6CYP1A2MAPTALDH1A1LMNA
SCHEMBL24253870 0.65 CYP2D6 (0.56) CYP2D6CYP1A2MAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022034587-A1 Traf2- AND Nck-INTERACTING KINASE (TNIK) INHIBITORS AND USES THEREOF TNIK THERAPEUTICS LTD (IL) 2022-02-17 WO disclosed