SCHEMBL24254494

SCHEMBL24254494

Cc1ccc(C(=O)NCc2ccccc2)cc1NC(=O)Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.55
LMNA P02545 2/20 0.53
PPARG P37231 5/20 0.53
ALDH1A1 P00352 2/20 0.53
HPGD P15428 1/20 0.53
HDAC1 Q13547 2/20 0.51
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HDAC4 P56524 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
HSD17B2 P37059 1/20 0.50
NR1H4 Q96RI1 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26188116 0.81 EPHX2 (0.61) EPHX2LMNAPPARGALDH1A1HPGD
SCHEMBL24254550 0.80 HPGD (0.46) LMNAALDH1A1HPGDCA1CA2
SCHEMBL24254499 0.79 LMNA (0.53) LMNAALDH1A1CA1CA2SMN1; SMN2
SCHEMBL27920895 0.79 EPHX2 (0.80) EPHX2PPARGALDH1A1HPGDHDAC1
SCHEMBL10323931 0.76 SMN1; SMN2 (0.63) EPHX2PPARGALDH1A1HPGDHDAC1
SCHEMBL24254507 0.74 MEN1 (0.48) LMNAALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL2971738 0.74 LMNA (0.66) EPHX2LMNAALDH1A1HPGDNR1H4
SCHEMBL24254503 0.74 MGAT2 (0.54) LMNAALDH1A1SMN1; SMN2MAPTHTT
SCHEMBL13947259 0.73 NR1H4 (0.80) LMNAALDH1A1HPGDHDAC1HDAC8
SCHEMBL3461067 0.73 EPHX2 (0.66) EPHX2LMNAPPARGALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230271918-A1 SUBSTITUTED 3-AMINO-4-METHYLBENZENESULFONAMIDES AS SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 DANA-FARBER CANCER INSTITUTE, INC. 2023-08-31 US disclosed
WO-2022035804-A1 SUBSTITUTED 3-AMINO-4-METHYLBENZENESULFONAMIDES AS SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230271918-A1 SUBSTITUTED 3-AMINO-4-METHYLBENZENESULFONAMIDES AS SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 USP28, USP30, USP1 EPHX2 4265/4885LMNA 3727/4885PPARG 4259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.