SCHEMBL2425936

SCHEMBL2425936

CCN(CC)c1ccc2c(c1)Sc1cc(N)c(Cc3ccccc3)cc1N2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100B P04271 1/20 0.37
CNR2 P34972 3/20 0.36
NOX1 Q9Y5S8 3/20 0.35
MAPK1 P28482 4/20 0.34
GAA P10253 4/20 0.34
MAPT P10636 4/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 4/20 0.33
TDP1 Q9NUW8 3/20 0.33
MEN1 O00255 3/20 0.33
HTT P42858 3/20 0.33
KMT2A Q03164 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
CDK2 P24941 1/20 0.33
TSHR P16473 2/20 0.33
NLRP3 Q96P20 1/20 0.32
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2429824 0.88 ADK (0.37) NOX1MAPK1GAAMAPTNPC1
SCHEMBL2429634 0.84 S100B (0.41) S100BNOX1MAPK1GAAMAPT
SCHEMBL2430499 0.82 S100B (0.38) S100BNOX1MAPK1GAAMAPT
SCHEMBL11763092 0.80 TSHR (0.54) CNR2NOX1MAPK1GAAMAPT
SCHEMBL972682 0.79 SNCA (0.46) S100BNOX1MAPK1GAAMAPT
SCHEMBL14321240 0.77 S100B (0.39) S100BNOX1MAPK1GAAMAPT
SCHEMBL2428865 0.77 SNCA (0.42) S100BNOX1MAPK1GAAMAPT
Iodide SCHEMBL3711619 0.77 NOX1 (0.55) CNR2NOX1MAPK1GAAMAPT
Iodide SCHEMBL3711622 0.77 NOX1 (0.55) CNR2NOX1MAPK1GAAMAPT
Iodide SCHEMBL3711621 0.77 NOX1 (0.55) CNR2NOX1MAPK1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547668-A1 TOLUIDINE BLUE DERIVATIVES AS PHOTOSENSITISING COMPOUNDS Pharmalucia Ltd (GB) 2013-01-23 EP disclosed
US-20120328530-A1 TOLUIDINE BLUE DERIVATIVES AS PHOTOSENSITISING COMPOUNDS PHARMALUCIA LIMITED (GB) 2012-12-27 US disclosed
WO-2011114137-A1 TOLUIDINE BLUE DERIVATIVES AS PHOTOSENSITISING COMPOUNDS PHARMALUCIA LIMITED (GB) 2011-09-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120328530-A1 TOLUIDINE BLUE DERIVATIVES AS PHOTOSENSITISING COMPOUNDS TYR, TST, TH S100B 1790/4885CNR2 1504/4885NOX1 635/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.