SCHEMBL242969

SCHEMBL242969

COc1cccc(C2c3ccc(O)cc3OCC2c2cccc(O)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.50
ESR2 Q92731 5/20 0.50
CYP19A1 P11511 2/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
ALOX12 P18054 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP3A4 P08684 2/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
MGAM O43451 1/20 0.40
EDNRB P24530 1/20 0.40
EDNRA P25101 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24103712 1.00 ESR1 (0.50) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL17965954 1.00 ESR1 (0.50) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL30362774 1.00 ESR1 (0.50) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL30362794 0.93 ESR1 (0.55) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL244280 0.93 ESR1 (0.55) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL24103707 0.93 ESR1 (0.55) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL17965956 0.93 ESR1 (0.55) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL28193659 0.92 CYP3A4 (0.49) ESR1ESR2CYP19A1MAPTMAPK1
SCHEMBL6092580 0.86 CYP3A4 (0.54) ESR1ESR2CYP19A1MAPTLMNA
SCHEMBL28194176 0.84 ESR1 (0.49) ESR1ESR2CYP19A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809618-B1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS INC (US) 2013-07-17 EP claimed
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-07-05 US claimed
US-8080675-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-20 US claimed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US claimed
US-12414934-B2 Combination therapies Aardvark Therapeutics, Inc. (US) 2025-09-16 US disclosed
WO-2024137472-A2 COMBINATION THERAPIES MEI PHARMA, INC. (US) 2024-06-27 WO disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
CN-116139125-A Combination therapy 梅制药公司 2023-05-23 CN disclosed
EP-4164632-A1 COMBINATION THERAPIES MEI Pharma, Inc. (US) 2023-04-19 EP disclosed
CN-107427003-B Combination therapy 梅制药公司 2023-01-31 CN disclosed
WO-2010045674-A1 METHODS FOR INDUCING PROGRAMMED CELL DEATH NOVOGEN RESEARCH PTY LTD (AU) 2010-04-29 WO disclosed
WO-2010022467-A1 IMMUNOMODULATING ACTIVITIES NOVOGEN RESEARCH PTY LTD (AU) 2010-03-04 WO disclosed
EP-2120925-A1 METHOD FOR INDUCING AUTOPHAGY Novogen Research Pty. Ltd. (AU) 2009-11-25 EP disclosed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP disclosed
WO-2008113100-A1 METHOD FOR INDUCING AUTOPHAGY NOVOGEN RESEARCH PTY LTD (AU) 2008-09-25 WO disclosed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP disclosed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US disclosed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414934-B2 Combination therapies PCK2, PDK1, PCK1 ESR1 2467/4885ESR2 1403/4885CYP19A1 3739/4885
US-20230233519-A1 COMBINATION THERAPIES BCL2, BAK1, BCL2L2 ESR1 3784/4885ESR2 2187/4885CYP19A1 2123/4885
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP19A1 2946/4885
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP19A1 2946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.