SCHEMBL24307129

SCHEMBL24307129

Clc1cccn2cc(-c3ccccc3)nc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A3 P47895 6/20 0.68
ALDH1A2 O94788 4/20 0.68
ALDH1A1 P00352 8/20 0.66
NPC1 O15118 7/20 0.66
RAB9A P51151 7/20 0.66
KDM4E B2RXH2 4/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
HSD17B10 Q99714 3/20 0.66
TP53 P04637 3/20 0.66
HPGD P15428 2/20 0.66
NPSR1 Q6W5P4 2/20 0.66
TSHR P16473 1/20 0.66
DHODH Q02127 1/20 0.59
PKM P14618 1/20 0.56
NFKB1 P19838 3/20 0.56
NFKB2 Q00653 3/20 0.56
RELA Q04206 3/20 0.56
MAPT P10636 2/20 0.56
PDE10A Q9Y233 1/20 0.55
ADORA1 P30542 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739105 0.85 RAB9A (0.68) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL5738406 0.85 ALDH1A1 (0.72) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL5738164 0.83 ALDH1A3 (0.51) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL4506816 0.82 RAB9A (0.56) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL5739101 0.82 RAB9A (0.52) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL5737395 0.82 PPARG (0.61) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL973108 0.81 ALDH1A3 (0.70) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL9082442 0.79 ALDH1A3 (0.68) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL4837433 0.79 ALDH1A1 (1.00) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A
SCHEMBL5737169 0.78 ALDH1A3 (0.50) ALDH1A3ALDH1A2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078306-A1 LARGE STERIC HINDERANCE PALLADIUM-NITROGEN-HETEROCYCLIC CARBENE COMPLEX, PREPARATION METHOD FOR SAME, APPLICATIONS OF SAME, AND SYNTHESIS METHOD FOR SONIDEGIB BASED ON SAME 中山大学 2022-04-21 WO disclosed