SCHEMBL24310314

SCHEMBL24310314

CONc1cccc(SNc2nc(Oc3c(C)cccc3Cl)cc(-c3ccccc3C)n2)c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.35
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPK14 Q16539 1/20 0.31
POLB P06746 2/20 0.31
SCN9A Q15858 1/20 0.31
USP2 O75604 1/20 0.31
BRD4 O60885 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24310579 0.92 RORC (0.35) RORCKDM4ELMNACYP1A2CYP2C19
SCHEMBL24309309 0.88 KDM4E (0.34) RORCKDM4ELMNACYP1A2CYP2C19
SCHEMBL24309263 0.87 POLB (0.34) KDM4ELMNAPOLBUSP2
SCHEMBL24310294 0.87 GPR39 (0.38) KDM4ELMNACYP1A2CYP2C19NPSR1
SCHEMBL24309707 0.84 PIK3CD (0.31) RORCKDM4ELMNACYP1A2CYP2C19
SCHEMBL24310302 0.80 BRD4 (0.37) RORCKDM4ELMNACYP1A2CYP2C19
SCHEMBL24309770 0.78 LMNA (0.34) LMNACYP1A2CYP2C19POLB
SCHEMBL24309252 0.77 RXRA (0.39) LMNANPSR1POLBMAPT
SCHEMBL24309777 0.74 LMNA (0.38) LMNACYP1A2CYP2C19NPSR1POLB
SCHEMBL24309507 0.72 CYP1A2 (0.35) LMNACYP1A2CYP2C19NPSR1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076627-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed