SCHEMBL2431240

SCHEMBL2431240

CC(C)(C)OC(=O)N1C[C@H](Oc2nccc3ccc(Br)cc23)C[C@@]1(C)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.35
GRM4 Q14833 4/20 0.33
USP30 Q70CQ3 2/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PLG P00747 1/20 0.32
PLAU P00749 1/20 0.32
PLAT P00750 1/20 0.32
CDK1 P06493 2/20 0.32
CCNB2 O95067 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
DGAT1 O75907 1/20 0.32
BACE1 P56817 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2428718 0.87 CYP3A4 (0.32) GRM4PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2430722 0.86 PIK3CD (0.38) GRM4PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL1244115 0.86 PIK3CD (0.47) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3302945 0.81 GPR119 (0.37) RORC
SCHEMBL2427449 0.81 PIK3CD (0.38) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL13433609 0.78 MCL1 (0.38) USP30PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL1273640 0.78 RXFP1 (0.42) RORC
SCHEMBL3305623 0.76 NCEH1 (0.40) RORC
SCHEMBL1072580 0.76 RAB9A (0.36) PIK3CDPIK3CAPIK3CBPIK3CGBACE1
SCHEMBL3302407 0.75 GPR119 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed