SCHEMBL24312409

SCHEMBL24312409

c1ccc(CCCNc2nnnc3ccccc23)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C19 P33261 1/20 1.00
GBA1 P04062 2/20 0.53
APP P05067 7/20 0.52
MAPK1 P28482 2/20 0.52
EGFR P00533 1/20 0.52
LMNA P02545 1/20 0.52
HTT P42858 1/20 0.52
PDE5A O76074 1/20 0.50
BCHE P06276 4/20 0.49
ACHE P22303 4/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HPGD P15428 1/20 0.47
PIK3CD O00329 1/20 0.47
PIK3R1 P27986 1/20 0.47
CASP6 P55212 1/20 0.47
KDM4E B2RXH2 1/20 0.46
JAK2 O60674 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24312413 0.81 CYP1A2 (0.68) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL3802400 0.80 CYP1A2 (0.67) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL8544714 0.79 APP (0.72) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL13948948 0.75 LMNA (0.81) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL4866885 0.74 GBA1 (0.59) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL4863010 0.72 GBA1 (0.58) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL4863857 0.72 PDE5A (0.82) GBA1MAPK1PDE5AKDM4EKMT2A
SCHEMBL4868696 0.72 LMNA (0.57) CYP1A2CYP2D6CYP2C19GBA1APP
SCHEMBL4865339 0.71 PDE5A (0.80) GBA1MAPK1PDE5AKDM4EKMT2A
SCHEMBL3636087 0.71 HRH4 (0.67) CYP1A2CYP2D6CYP2C19MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11732286-B2 T5 exonuclease-based method to identify DNA topoisomerase inhibitors THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2023-08-22 US disclosed
US-11732286-B2 T5 exonuclease-based method to identify DNA topoisomerase inhibitors THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2023-08-22 US disclosed
US-20220170070-A1 T5 EXONUCLEASE-BASED METHOD TO IDENTIFY DNA TOPOISOMERASE INHIBITORS THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2022-06-02 US disclosed
US-20220119858-A1 T5 EXONUCLEASE-BASED METHOD TO IDENTIFY DNA TOPOISOMERASE INHIBITORS THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2022-04-21 US disclosed
US-11268129-B1 T5 exonuclease-based method to identify DNA topoisomerase inhibitors THE FLORIDA INTERNATIONAL UNIVERSITY BOARD OF TRUSTEES (US) 2022-03-08 US disclosed