SCHEMBL24313723

SCHEMBL24313723

CC(C)c1ccc(OCC2CC2)c(SCl)c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.38
PDE4A P27815 3/20 0.38
PDE4C Q08493 3/20 0.38
PDE4D Q08499 3/20 0.38
KMO O15229 1/20 0.37
RIPK1 Q13546 1/20 0.35
ACACB O00763 4/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
DHFR P00374 1/20 0.35
GRM2 Q14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24313917 0.86 PDE4B (0.38) PDE4BPDE4APDE4CPDE4DRIPK1
SCHEMBL24314212 0.81 ACACB (0.39) ACACB
SCHEMBL13678313 0.81 KMO (0.47) PDE4BPDE4APDE4CPDE4DKMO
SCHEMBL16852267 0.79 PDE4B (0.43) PDE4BPDE4APDE4CPDE4DRIPK1
SCHEMBL13678365 0.78 XDH (0.48) PDE4B
SCHEMBL18120363 0.78 TRPV1 (0.45) PDE4BPDE4APDE4CPDE4D
SCHEMBL24313901 0.78 DHFR (0.44) PDE4BPDE4APDE4CPDE4DRIPK1
SCHEMBL11951596 0.78 ACACB (0.45) PDE4BPDE4APDE4CPDE4DRIPK1
SCHEMBL1438963 0.78 NPC1 (0.50) PDE4BPDE4APDE4CPDE4DRIPK1
SCHEMBL24314286 0.75 HTR2C (0.38) PDE4BPDE4APDE4CPDE4DKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed
WO-2022081807-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed