SCHEMBL24313817

SCHEMBL24313817

COC(=O)c1ccc(Oc2cnc3cc(Br)ccc3c2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
HPGDS O60760 5/20 0.42
THRB P10828 1/20 0.42
MAPK1 P28482 2/20 0.42
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP13 P45452 1/20 0.41
HTT P42858 2/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
GABRA5 P31644 1/20 0.39
PDE4B Q07343 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24313800 0.87 LMNA (0.46) LMNAHPGDSMAPK1HTTL3MBTL1
SCHEMBL2001821 0.82 HPGDS (0.51) HPGDSMAPK1MMP2MMP9MMP8
SCHEMBL24313798 0.79 LIPE (0.43) LMNAHPGDSMAPK1PDE4BSCN9A
SCHEMBL21838860 0.76 LMNA (0.65) LMNAMAPK1TSHRL3MBTL1KDM4E
SCHEMBL23474086 0.76 LMNA (0.52) LMNAMAPK1TSHRL3MBTL1KDM4E
SCHEMBL30617764 0.74 HTT (0.52) HPGDSMAPK1MMP2MMP9MMP8
SCHEMBL25255029 0.74 HTT (0.52) HPGDSMAPK1MMP2MMP9MMP8
SCHEMBL23474167 0.74 LMNA (0.41) LMNATHRBMAPK1MMP2MMP9
SCHEMBL4596324 0.73 LMNA (0.52) LMNAMAPK1TSHRL3MBTL1KDM4E
SCHEMBL3586183 0.73 LMNA (0.60) LMNAMAPK1TSHRL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022077161-A1 COMPOUNDS FOR MODULATING ACTIVITY OF FXR AND USES THEREOF GANNEX PHARMA CO., LTD. (CN) 2022-04-21 WO disclosed
CN-114315815-A Compounds for modulating FXR activity and uses thereof 甘莱制药有限公司 2022-04-12 CN disclosed