SCHEMBL24316549

SCHEMBL24316549

COc1ccc(CCOc2ncc(Oc3ccc4ncc(C)c(=O)n4c3)cc2OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 2/20 0.43
RXFP1 Q9HBX9 1/20 0.38
PIK3CA P42336 4/20 0.38
MTOR P42345 3/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
PDE1A P54750 2/20 0.34
PDE1B Q01064 2/20 0.34
PDE1C Q14123 2/20 0.34
GRM2 Q14416 1/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
POLB P06746 1/20 0.34
P2RX7 Q99572 1/20 0.33
NPBWR1 P48145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316622 0.94 CYP11B1 (0.39) CSF1RRXFP1PIK3CAMTORCYP11B1
SCHEMBL24316620 0.91 CSF1R (0.37) CSF1RRXFP1PIK3CAMTORALDH1A1
SCHEMBL24316434 0.90 CSF1R (0.53) CSF1RRXFP1PIK3CAMTORKDM4E
SCHEMBL24316621 0.87 PIK3CA (0.38) CSF1RRXFP1PIK3CAMTORKDM4E
SCHEMBL24316982 0.86 CSF1R (0.48) CSF1RRXFP1PIK3CAMTORKDM4E
SCHEMBL24316814 0.84 CSF1R (0.47) CSF1RRXFP1PIK3CAMTORKDM4E
SCHEMBL24316983 0.84 CSF1R (0.46) CSF1RRXFP1PIK3CAMTORALDH1A1
SCHEMBL24316448 0.83 CSF1R (0.45) CSF1RRXFP1PIK3CAMTORPDE1A
SCHEMBL24316545 0.82 CSF1R (0.43) CSF1RRXFP1PIK3CAMTORKDM4E
SCHEMBL24316661 0.82 CSF1R (0.52) CSF1RRXFP1PIK3CAMTORPDE1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed