SCHEMBL24316434

SCHEMBL24316434

COc1ccc(COc2ncc(Oc3ccc4ncc(C)c(=O)n4c3)cc2OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 4/20 0.53
PIK3CA P42336 5/20 0.39
MTOR P42345 4/20 0.39
RXFP1 Q9HBX9 1/20 0.37
ALKBH1 Q13686 1/20 0.37
GRM5 P41594 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
KIT P10721 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316982 0.95 CSF1R (0.48) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316814 0.93 CSF1R (0.47) CSF1RPIK3CAMTORRXFP1GRM5
SCHEMBL24316983 0.93 CSF1R (0.46) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316545 0.92 CSF1R (0.43) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316448 0.92 CSF1R (0.45) CSF1RPIK3CAMTORRXFP1GRM5
SCHEMBL24316565 0.91 CSF1R (0.44) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316661 0.91 CSF1R (0.52) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316437 0.91 CSF1R (0.45) CSF1RPIK3CAMTORRXFP1ALKBH1
SCHEMBL24316549 0.90 CSF1R (0.43) CSF1RPIK3CAMTORRXFP1KDM4E
SCHEMBL24316587 0.90 CSF1R (0.44) CSF1RPIK3CAMTORRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed