SCHEMBL2431765

SCHEMBL2431765

O=C(O)c1cc(Oc2ccc(-n3ccnc3)cc2)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 4/20 0.50
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 2/20 0.46
ICAM1 P05362 2/20 0.46
SELE P16581 2/20 0.46
VCAM1 P19320 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP19A1 P11511 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
BAZ2B Q9UIF8 1/20 0.46
NOS2 P35228 3/20 0.46
PORCN Q9H237 1/20 0.46
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
ALDH1A1 P00352 1/20 0.44
ENPP2 Q13822 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364087 0.81 ADH5 (0.75) ADH5CYP3A4HTTBAZ2BHTR2A
SCHEMBL22437049 0.81 ADH5 (0.53) ADH5CYP3A4CYP19A1HTTBAZ2B
SCHEMBL30900589 0.81 ADH5 (0.53) ADH5CYP3A4CYP19A1HTTBAZ2B
SCHEMBL10512975 0.78 LMNA (0.62) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL21940149 0.76 CYP3A4 (0.62) ADH5CYP3A4CYP2D6ICAM1SELE
SCHEMBL4365227 0.76 KDM4E (0.49) ALDH1A1
SCHEMBL22737610 0.76 GCK (0.54) ALDH1A1
SCHEMBL7005980 0.76 CYP3A4 (0.69) CYP3A4CYP2D6CYP1A2CYP19A1CYP2C9
SCHEMBL4334161 0.75 ALDH1A1 (0.47) CYP3A4ALDH1A1
SCHEMBL2427202 0.75 P2RX3 (0.52) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011117254-A1 PIPERIDINE AMIDES AS MODULATORS OF THE GHRELIN RECEPTOR PROSIDION LIMITED (GB) 2011-09-29 WO disclosed