SCHEMBL24323744

SCHEMBL24323744

O=Cc1ncc(N2CCOCC2)cc1N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 1/20 0.44
ALDH1A3 P47895 1/20 0.44
LGMN Q99538 2/20 0.44
PIK3CD O00329 2/20 0.43
PIK3CA P42336 2/20 0.43
PIK3CB P42338 2/20 0.43
PIK3CG P48736 1/20 0.43
PRKDC P78527 1/20 0.43
POLB P06746 1/20 0.42
MAPT P10636 4/20 0.41
ALDH1A1 P00352 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DHFR P00374 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
AKR1C3 P42330 1/20 0.39
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24323225 0.83 ALDH1A1 (0.46) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL18989023 0.83 ALDH3A1 (0.50) ALDH3A1ALDH1A3PRKDCMAPTALDH1A1
SCHEMBL359690 0.76 LGMN (0.56) LGMNPIK3CDPIK3CAPIK3CBPOLB
SCHEMBL24323360 0.75 POLB (0.47) ALDH3A1ALDH1A3PIK3CDPIK3CAPIK3CB
SCHEMBL3646284 0.73 ALDH1A1 (0.48) ALDH3A1ALDH1A3PIK3CDPIK3CAPIK3CB
SCHEMBL361410 0.73 POLB (0.57) POLBMAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL6224618 0.71 PIK3CD (0.69) ALDH3A1ALDH1A3LGMNPIK3CDPIK3CA
SCHEMBL98667 0.71 ALDH3A1 (0.46) ALDH3A1ALDH1A3PIK3CDPIK3CAPIK3CB
SCHEMBL3645584 0.71 MAPT (0.58) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL18412831 0.70 ALDH1A1 (0.46) LGMNPRKDCPOLBMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4225765-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR Vertex Pharmaceuticals Incorporated (US) 2023-08-16 EP disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed