SCHEMBL24325433

SCHEMBL24325433

Cc1cccc(C)c1-c1cc(Cl)nc(NSc2cccc(C(=O)N3CCN(C(=O)OC(C)(C)C)CC(O)C3)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.37
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
USP30 Q70CQ3 2/20 0.34
CCNK O75909 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCND3 P30281 1/20 0.33
CDK9 P50750 1/20 0.33
CDK6 Q00534 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CRBN Q96SW2 1/20 0.33
IDH1 O75874 1/20 0.33
RHOA P61586 1/20 0.33
POLB P06746 1/20 0.33
PARP14 Q460N5 1/20 0.33
BTK Q06187 1/20 0.32
ROCK2 O75116 1/20 0.32
SMARCA2 P51531 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326078 1.00 EPHX2 (0.37) EPHX2MEN1KMT2AUSP30CCNK
SCHEMBL24326398 0.97 MEN1 (0.37) EPHX2MEN1KMT2AUSP30HSP90AA1
SCHEMBL24326125 0.87 RHOA (0.32) MEN1KMT2ARHOAPOLB
SCHEMBL24325763 0.86 MMP3 (0.32)
SCHEMBL24326520 0.86 PARP1 (0.33) EPHX2
SCHEMBL24326178 0.86 MMP3 (0.32)
SCHEMBL24326259 0.86 PARP1 (0.33) EPHX2
SCHEMBL24326087 0.84 TGFBR1 (0.43) KMT2APOLB
SCHEMBL24326268 0.84 TGFBR1 (0.43) KMT2APOLB
SCHEMBL29570536 0.84 TGFBR1 (0.43) KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed