SCHEMBL24326398

SCHEMBL24326398

Cc1cccc(C)c1-c1cc(Cl)nc(NSc2cccc(C(=O)N3CCCN(C(=O)OC(C)(C)C)CC(O)C3)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
USP30 Q70CQ3 1/20 0.36
RHOA P61586 2/20 0.35
EPHX2 P34913 1/20 0.35
ANO1 Q5XXA6 1/20 0.33
TP53 P04637 1/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 2/20 0.33
PARP1 P09874 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
BTK Q06187 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
PIM1 P11309 2/20 0.32
PIM2 Q9P1W9 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326078 0.97 EPHX2 (0.37) MEN1KMT2AUSP30RHOAEPHX2
SCHEMBL24325433 0.97 EPHX2 (0.37) MEN1KMT2AUSP30RHOAEPHX2
SCHEMBL24325763 0.85 MMP3 (0.32) TRPV3
SCHEMBL24326178 0.85 MMP3 (0.32) TRPV3
SCHEMBL29570518 0.85 TGFBR1 (0.42) KMT2A
SCHEMBL24326411 0.85 TGFBR1 (0.42) KMT2A
SCHEMBL24326125 0.84 RHOA (0.32) MEN1KMT2ARHOA
SCHEMBL24326520 0.83 PARP1 (0.33) EPHX2PARP1TRPV3
SCHEMBL24326259 0.83 PARP1 (0.33) EPHX2PARP1TRPV3
SCHEMBL24326268 0.81 TGFBR1 (0.43) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed