SCHEMBL24325812

SCHEMBL24325812

Cc1cccc(C)c1-c1cc(O)nc(NSc2cccc(N3CCCN(C)CC3)c2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 2/20 0.39
LCK P06239 2/20 0.37
ADRA2C P18825 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
CDK2 P24941 5/20 0.35
CCNA2 P20248 2/20 0.35
CDK9 P50750 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
CCNK O75909 1/20 0.35
CCND3 P30281 1/20 0.35
CDK6 Q00534 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
FLT3 P36888 3/20 0.34
KIT P10721 2/20 0.34
PLK4 O00444 1/20 0.34
CHEK1 O14757 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24325710 0.86 HRH3 (0.31)
SCHEMBL24326123 0.85 CYBB (0.33)
SCHEMBL24326318 0.85 DRD2 (0.44)
SCHEMBL24325712 0.83
SCHEMBL24326652 0.83 FFAR4 (0.32)
SCHEMBL24325715 0.83 FFAR4 (0.32)
SCHEMBL24325821 0.83 GPR119 (0.41) JAK2JAK3CDK2CCNA2CDK9
SCHEMBL24326648 0.82 GAA (0.32)
SCHEMBL24326270 0.82 FFAR4 (0.32)
SCHEMBL24326160 0.82 NR1I2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed