SCHEMBL24326318

SCHEMBL24326318

Cc1cccc(C)c1-c1cc(O)nc(NSc2cccc(N3CCCN(Cc4ccccc4)CC3)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.44
DRD3 P35462 1/20 0.44
DRD4 P21917 2/20 0.38
SCN9A Q15858 1/20 0.37
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
USP2 O75604 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
XBP1 P17861 1/20 0.36
KMT2A Q03164 1/20 0.36
CASP1 P29466 1/20 0.36
CASP5 P51878 1/20 0.36
CYBB P04839 1/20 0.36
NOX4 Q9NPH5 1/20 0.36
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326123 0.87 CYBB (0.33) DRD2MAPTXBP1CYBBNOX4
SCHEMBL24325812 0.85 MAP4K1 (0.39)
SCHEMBL24325710 0.82 HRH3 (0.31)
SCHEMBL24326315 0.82 SIGMAR1 (0.39) DRD2DRD3DRD4HTR3EHTR3B
SCHEMBL24325712 0.78
SCHEMBL24325715 0.78 FFAR4 (0.32)
SCHEMBL24326652 0.78 FFAR4 (0.32)
SCHEMBL24325821 0.78 GPR119 (0.41) MAPTMEN1KMT2A
SCHEMBL24326648 0.78 GAA (0.32)
SCHEMBL24326270 0.78 FFAR4 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed