SCHEMBL2432899

SCHEMBL2432899

CCC(C(=O)O)c1ccc(NC(=O)c2nccc3ccccc23)c(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
FLT3 P36888 1/20 0.41
ITGB1 P05556 2/20 0.40
ITGA4 P13612 2/20 0.40
CNR2 P34972 2/20 0.39
GAA P10253 2/20 0.39
NPC1 O15118 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CCR1 P32246 1/20 0.39
AKR1C3 P42330 4/20 0.39
AKR1C2 P52895 4/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91549 0.80 RAB9A (0.62) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL2433435 0.78 RAB9A (0.50) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL14626752 0.77 MAPT (0.47) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL14591892 0.77 MAPT (0.44) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL12327918 0.76 MEN1 (0.47) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL2432847 0.76 ITGB1 (0.46) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL14491714 0.75 ITGB1 (0.46) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL27578589 0.75 KMT2A (0.44) RAB9AMAPTMEN1KMT2ATP53
SCHEMBL2432438 0.75 NPC1 (0.48) MAPTMEN1KMT2ANPC1ALDH1A1
SCHEMBL2429653 0.74 AKR1B1 (0.46) RAB9AMAPTMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1346982-B1 VLA-4 INHIBITORS DAIICHI SEIYAKU CO (JP) 2011-09-14 EP disclosed