SCHEMBL24330613

SCHEMBL24330613

Cc1ncc(N2CC[C@@](C)(I)C2)cn1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
CHRNA4 P43681 2/20 0.34
OPRL1 P41146 1/20 0.31
CHRNA1 P02708 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30
CHRNA7 P36544 1/20 0.30
CHRND Q07001 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24324476 0.82 SIGMAR1 (0.36) CHRNB2CHRNB4CHRNA3CHRNA4OPRL1
SCHEMBL23561133 0.71 CDK4 (0.40) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL20468861 0.70 ALDH1A1 (0.50)
SCHEMBL23228760 0.69 TSHR (0.34) OPRL1
SCHEMBL12204161 0.69 CHKA (0.43) CHRNB2CHRNA4
SCHEMBL9881482 0.67 MAPT (0.44) CHRNB2CHRNA4
SCHEMBL8281056 0.66 HTR3A (0.50)
SCHEMBL20311310 0.64 CHRNB2 (0.59) CHRNB2CHRNA4
SCHEMBL22361873 0.64 CHRNB2 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL15706151 0.64 POLB (0.39) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076620-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed