SCHEMBL24337073

SCHEMBL24337073

COC(=O)C12CC(C1)C(NC(=O)OC(C)(C)C)C2

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 7/20 0.49
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
KDM1A O60341 1/20 0.37
BTK Q06187 1/20 0.37
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
GAA P10253 1/20 0.36
CTSK P43235 2/20 0.35
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23562416 1.00 HSD11B1 (0.49) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL23900563 0.86 BTK (0.44) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL24543130 0.86 BTK (0.44) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL23625485 0.86 BTK (0.44) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL26014913 0.84 HSD11B1 (0.48) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL26014916 0.82 HSD11B1 (0.39) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL23281289 0.78 NFKB1 (0.40) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL23562417 0.76 HSD11B1 (0.47) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL24701274 0.75 HSD11B1 (0.48) HSD11B1NFKB1NFKB2RELAKDM1A
SCHEMBL23161367 0.74 HSD11B1 (0.40) HSD11B1MEN1MAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023150291-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF USE SCHRÖDINGER, INC. (US) 2023-08-10 WO disclosed
WO-2023081662-A1 BICYCLIC DERIVATIVES AS CCR2 MODULATORS ARIA PHARMACEUTICALS, INC. (US) 2023-05-11 WO disclosed
WO-2022066864-A1 SHMT INHIBITORS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2022-03-31 WO disclosed
US-9586978-B2 Anti-viral compounds ABBVIE INC. (US) 2017-03-07 US disclosed