SCHEMBL24344900

SCHEMBL24344900

Cc1cnc2c(c1)C1C[C@H]1N2

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
PDK2 Q15119 1/20 0.31
PDK4 Q16654 1/20 0.31
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
NNMT P40261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20124978 0.84 DRD2 (0.35) CHRNB2CHRNA4DRD2DRD1PDK2
SCHEMBL20125119 0.84 DRD2 (0.35) CHRNB2CHRNA4DRD2DRD1PDK2
SCHEMBL23938075 0.72 CHRNB2 (0.31) CHRNB2CHRNA4
SCHEMBL23416751 0.67
SCHEMBL13199592 0.66 CA1 (0.36) CHRNB2CHRNA4DRD2DRD1PDK2
SCHEMBL7914307 0.66 CA1 (0.36) CHRNB2CHRNA4DRD2DRD1PDK2
SCHEMBL7921085 0.63 CCR1 (0.32) CCR1CCR5CCR8NOS3NOS1
SCHEMBL7914306 0.62 NNMT (0.58) CCR1CCR5CCR8NOS3NOS1
SCHEMBL21729487 0.62 NNMT (0.58) CCR1CCR5CCR8NOS3NOS1
SCHEMBL13330178 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076975-A1 5- AND 6-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ENLIVEN THERAPEUTICS, INC. (US) 2022-04-14 WO disclosed