SCHEMBL24359488

SCHEMBL24359488

NC(=O)CCCCCCSC(=O)CCc1cccc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 10/20 0.54
TAAR1 Q96RJ0 1/20 0.51
AURKA O14965 2/20 0.46
NR3C2 P08235 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
FFAR1 O14842 2/20 0.44
FFAR4 Q5NUL3 2/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30412030 0.85 EPHX1 (0.59) EPHX1TAAR1AURKANR3C2HDAC1
SCHEMBL249437 0.84 EPHX1 (0.61) EPHX1TAAR1AURKANR3C2HDAC1
SCHEMBL185922 0.84 TAAR1 (0.62) EPHX1TAAR1AURKANR3C2HDAC1
SCHEMBL30645023 0.84 TAAR1 (0.62) EPHX1TAAR1AURKANR3C2HDAC1
SCHEMBL24359482 0.83 TAAR1 (0.47) TAAR1NR3C2FFAR1
SCHEMBL4309679 0.82 TAAR1 (0.60) EPHX1TAAR1AURKANR3C2HDAC1
SCHEMBL24359351 0.80 NOS1 (0.50) HDAC1HDAC8FFAR1
SCHEMBL8491974 0.75 TAAR1 (0.61) EPHX1TAAR1NR3C2HDAC1HDAC8
SCHEMBL7150587 0.74 MAPT (0.60) EPHX1TAAR1HDAC1HDAC8FFAR1
SCHEMBL24359478 0.74 FFAR1 (0.42) EPHX1TAAR1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022087456-A1 NEW COMPOUNDS FOR THE TREATMENT OF ALZHEIMER'S DISEASE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-04-28 WO disclosed