SCHEMBL4309679

SCHEMBL4309679

NC(=O)CCCc1cccc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.60
EPHX1 P07099 6/20 0.58
HDAC1 Q13547 1/20 0.58
HDAC8 Q9BY41 1/20 0.58
AURKA O14965 2/20 0.57
NR3C2 P08235 1/20 0.54
ATM Q13315 1/20 0.52
ACP3 P15309 1/20 0.51
MAOB P27338 1/20 0.51
IDO1 P14902 1/20 0.50
GRM2 Q14416 1/20 0.49
GRM3 Q14832 1/20 0.49
FFAR1 O14842 2/20 0.49
FFAR4 Q5NUL3 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249437 0.95 EPHX1 (0.61) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL30412030 0.94 EPHX1 (0.59) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL185922 0.92 TAAR1 (0.62) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL30645023 0.92 TAAR1 (0.62) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL1981615 0.87 FFAR4 (0.59) TAAR1EPHX1HDAC1HDAC8ACP3
SCHEMBL27930024 0.86 HDAC1 (0.57) TAAR1EPHX1HDAC1HDAC8NR3C2
SCHEMBL18798841 0.85 HDAC1 (0.71) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL11755472 0.83 HDAC1 (0.60) TAAR1EPHX1HDAC1HDAC8ACP3
SCHEMBL24359488 0.82 EPHX1 (0.54) TAAR1EPHX1HDAC1HDAC8AURKA
SCHEMBL28673196 0.82 LMNA (0.60) TAAR1EPHX1HDAC1HDAC8NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN claimed
CN-101495458-B Substituted arylimidazolone and triazolone as inhibitors of vasopressin receptors BAYER IP GMBH 2014-01-29 CN disclosed
WO-2009137338-A1 PYRAZOLE COMPOUNDS AS CCR1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-11-12 WO disclosed
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN disclosed