SCHEMBL24377993

SCHEMBL24377993

NC(=O)C1CN(C(=O)CCl)c2cc(Br)ccc2O1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 16/20 0.49
SIRT2 Q8IXJ6 11/20 0.49
CASP2 P42575 1/20 0.45
POLB P06746 1/20 0.41
SIRT3 Q9NTG7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29516214 1.00 SIRT1 (0.49) SIRT1SIRT2CASP2POLBSIRT3
SCHEMBL24378120 0.90 SIRT1 (0.47) SIRT1SIRT2CASP2SIRT3
SCHEMBL26938747 0.89 CASP2 (0.47) SIRT1SIRT2CASP2POLB
SCHEMBL29516124 0.85 TP53 (0.49) SIRT1POLB
SCHEMBL24378122 0.85 TP53 (0.49) SIRT1POLB
SCHEMBL24378019 0.83 SIRT1 (0.48) SIRT1SIRT2POLBSIRT3
SCHEMBL26938829 0.83 SIRT1 (0.65) SIRT1SIRT2SIRT3
SCHEMBL24378118 0.83 SIRT1 (0.65) SIRT1SIRT2SIRT3
SCHEMBL24378125 0.83 SIRT1 (0.65) SIRT1SIRT2SIRT3
SCHEMBL24378126 0.80 SIRT1 (0.56) SIRT1SIRT2POLBSIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230399304-A1 COVALENT INHIBITORS OF CREATINE KINASE (CK) AND USES THEREOF FOR TREATING AND PREVENTING CANCER DANA-FARBER CANCER INSTITUTE, INC. 2023-12-14 US disclosed
US-20230399304-A1 COVALENT INHIBITORS OF CREATINE KINASE (CK) AND USES THEREOF FOR TREATING AND PREVENTING CANCER DANA-FARBER CANCER INSTITUTE, INC. 2023-12-14 US disclosed
CN-116323571-A Covalent inhibitors of Creatine Kinase (CK) and their use for the treatment and prevention of cancer 丹娜法伯癌症研究院 2023-06-23 CN disclosed
WO-2022087433-A1 COVALENT INHIBITORS OF CREATINE KINASE (CK) AND USES THEREOF FOR TREATING AND PREVENTING CANCER DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-04-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230399304-A1 COVALENT INHIBITORS OF CREATINE KINASE (CK) AND USES THEREOF FOR TREATING AND PREVENTING CANCER CKMT1A; CKMT1B, PHKG1, PCK1 SIRT1 935/4885SIRT2 1211/4885CASP2 941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.