SCHEMBL24378463

SCHEMBL24378463

Cc1csc(-c2cc[nH]n2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.50
CYP3A4 P08684 2/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
SRC P12931 1/20 0.39
CDK2 P24941 1/20 0.39
ZAP70 P43403 1/20 0.39
SYK P43405 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
NOS1 P29475 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29438488 0.81 CYP19A1 (0.37) CYP3A4KDM4EALDH1A1HPGDMEN1
SCHEMBL31341048 0.73 RAB9A (0.57) KDM4EALDH1A1MEN1MAPK1KMT2A
SCHEMBL13377800 0.72 PDE10A (0.67) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL18157874 0.72 SMN1; SMN2 (0.55) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL24378644 0.72 ECE1 (0.42) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL30574726 0.70 PDE10A (0.46) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL8198560 0.69 CYP3A4 (0.60) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL6840531 0.68 PDE10A (0.52) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL7905176 0.67 CYP3A4 (0.58) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL1673128 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036718-A ALK5 inhibitor and preparation method and application thereof 安炎达医药技术(广州)有限公司 2026-05-15 CN disclosed
WO-2022086993-A1 NOVEL INHIBITORS OF PIKFYVE AND METHODS USING SAME TME THERAPEUTICS LLC (US) 2022-04-28 WO disclosed
CN-1046275-C 2-methoxyiminophenyl-N-methylacetamide derivatives, process for their preparation, their use and compositions containing them BASF AG (DE) 1999-11-10 CN disclosed
CN-1118165-A Ortho-substituted 2-methoxyiminophenylacetic acid methylamides BASF AG (DE) 1996-03-06 CN disclosed