SCHEMBL24417455

SCHEMBL24417455

O=Cc1cc(Br)ccc1-c1nnn[nH]1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.42
CYP2A6 P11509 2/20 0.37
PTPN1 P18031 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
XDH P47989 1/20 0.33
GPR35 Q9HC97 7/20 0.33
PIM3 Q86V86 2/20 0.32
S100A4 P26447 1/20 0.32
PIM1 P11309 1/20 0.31
TGM2 P21980 1/20 0.30
CES1 P23141 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24416785 0.88 ERN1 (0.39) ERN1CYP2A6PTPN1PTGDR2XDH
SCHEMBL3633061 0.81 XDH (0.51) ERN1PTPN1XDHS100A4TGM2
SCHEMBL1647011 0.77 XDH (0.46) CYP2A6XDHALDH1A1
SCHEMBL1629842 0.76 ALOX5AP (0.36) GPR35S100A4
SCHEMBL10254523 0.76 GPR35 (0.35) GPR35S100A4
SCHEMBL203395 0.75 ERN1 (0.61) ERN1CYP2A6PTPN1PTGDR2PIM3
SCHEMBL2838019 0.72 IDO1 (0.57) GPR35TGM2CES1ALDH1A1
SCHEMBL30192181 0.72 IDO1 (0.57) GPR35TGM2CES1ALDH1A1
SCHEMBL24416831 0.72 DYRK1A (0.33) XDHALDH1A1
SCHEMBL24416917 0.72 KCNJ1 (0.34) ERN1PTPN1XDHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022095965-A1 TETRAZOLE DERIVATIVE, PREPARATION FOR TETRAZOLE DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING TETRAZOLE DERIVATIVE, AND APPLICATION OF TETRAZOLE DERIVATIVE 浙江大学 2022-05-12 WO disclosed