SCHEMBL244269

SCHEMBL244269

Oc1ccc(C2COc3cc(O)ccc3C2c2ccccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.64
ESR2 Q92731 7/20 0.64
CYP3A4 P08684 1/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27288519 1.00 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL24103708 1.00 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL30362800 1.00 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL24103716 1.00 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL2717066 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL10074006 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL30362812 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL243810 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL21613691 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL18898251 0.94 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809618-B1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS INC (US) 2013-07-17 EP claimed
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-07-05 US claimed
US-8080675-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-20 US claimed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP claimed
CN-101094844-A Chroman derivatives, medicaments and use in therapy NOVOGEN RES PTY LTD (AU) 2007-12-26 CN claimed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP claimed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US claimed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO claimed
US-12414934-B2 Combination therapies Aardvark Therapeutics, Inc. (US) 2025-09-16 US disclosed
WO-2024137472-A2 COMBINATION THERAPIES MEI PHARMA, INC. (US) 2024-06-27 WO disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
CN-116139125-A Combination therapy 梅制药公司 2023-05-23 CN disclosed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP disclosed
WO-2008113100-A1 METHOD FOR INDUCING AUTOPHAGY NOVOGEN RESEARCH PTY LTD (AU) 2008-09-25 WO disclosed
CN-101094844-A Chroman derivatives, medicaments and use in therapy NOVOGEN RES PTY LTD (AU) 2007-12-26 CN disclosed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP disclosed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US disclosed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414934-B2 Combination therapies PCK2, PDK1, PCK1 ESR1 2467/4885ESR2 1403/4885CYP3A4 4003/4885
US-20230233519-A1 COMBINATION THERAPIES BCL2, BAK1, BCL2L2 ESR1 3784/4885ESR2 2187/4885CYP3A4 4039/4885
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP3A4 1392/4885
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP3A4 1392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.