SCHEMBL243810

SCHEMBL243810

Oc1ccc(C2COc3cc(O)ccc3C2c2ccc(O)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.57
ESR2 Q92731 7/20 0.57
CYP3A4 P08684 1/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
TTR P02766 1/20 0.49
ALOX15B O15296 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362812 1.00 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL2717066 1.00 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL18898251 1.00 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL10074006 1.00 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL21613691 1.00 ESR1 (0.57) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL24103716 0.94 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL30362800 0.94 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL24103708 0.94 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL244269 0.94 ESR1 (0.64) ESR1ESR2CYP3A4MAOAMAOB
SCHEMBL24103714 0.93 ESR2 (0.52) ESR1ESR2CYP3A4MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 162 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140234295-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2014-08-21 US claimed
US-20130273177-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2013-10-17 US claimed
EP-1809618-B1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS INC (US) 2013-07-17 EP claimed
US-20120251630-A1 REMISSION THERAPY OF CANCER WITH ISOFLAVONOIDS MARSHALL EDWARDS, INC. (US) 2012-10-04 US claimed
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-07-05 US claimed
US-8163795-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2012-04-24 US claimed
US-20120039917-A1 IMMUNOMODULATING ACTIVITIES MARSHALL EDWARDS, INC. 2012-02-16 US claimed
US-20120004296-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC (US) 2012-01-05 US claimed
US-8080675-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-20 US claimed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP claimed
CN-101094844-A Chroman derivatives, medicaments and use in therapy NOVOGEN RES PTY LTD (AU) 2007-12-26 CN claimed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP claimed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US claimed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO claimed
US-12414934-B2 Combination therapies Aardvark Therapeutics, Inc. (US) 2025-09-16 US disclosed
US-12329739-B2 Isoflavonoid compounds and methods for the treatment of cancer Aardvark Therapeutic, Inc. (US) 2025-06-17 US disclosed
US-12318364-B2 Isoflavonoid compositions and methods for the treatment of cancer Aardvark Therapeutics, Inc. (US) 2025-06-03 US disclosed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP disclosed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US disclosed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414934-B2 Combination therapies PCK2, PDK1, PCK1 ESR1 2467/4885ESR2 1403/4885CYP3A4 4003/4885
US-20120251630-A1 REMISSION THERAPY OF CANCER WITH ISOFLAVONOIDS CYP19A1, HSD17B11, BRCA1 ESR1 71/4885ESR2 9/4885CYP3A4 983/4885
US-20120039917-A1 IMMUNOMODULATING ACTIVITIES CD4, NFATC1, HRH2 ESR1 138/4885ESR2 43/4885CYP3A4 1056/4885
US-20130273177-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, SI ESR1 176/4885ESR2 154/4885CYP3A4 683/4885
US-12318364-B2 Isoflavonoid compositions and methods for the treatment of cancer BAX, CASP3, SI ESR1 176/4885ESR2 154/4885CYP3A4 683/4885
US-20140234295-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, API5 ESR1 57/4885ESR2 22/4885CYP3A4 2283/4885
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP3A4 1392/4885
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP3A4 1392/4885
US-20120004296-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885CYP3A4 1392/4885
US-12329739-B2 Isoflavonoid compounds and methods for the treatment of cancer BAX, CASP3, API5 ESR1 57/4885ESR2 22/4885CYP3A4 2283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.