SCHEMBL2443409

SCHEMBL2443409

CC(C)Oc1c(Cl)cc(-c2csc(NC(=O)CBr)n2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 7/20 0.47
MAPT P10636 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
PI4KB Q9UBF8 1/20 0.46
TRPA1 O75762 2/20 0.46
XIAP P98170 1/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CLK1 P49759 1/20 0.43
USP2 O75604 1/20 0.43
CASP3 P42574 1/20 0.42
SENP7 Q9BQF6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2453828 0.93 ABL1 (0.48) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL4410358 0.89 ABL1 (0.47) ABL1MAPTPI4KBTRPA1ROCK2
SCHEMBL480411 0.87 TRPA1 (0.58) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL2443035 0.85 MAPT (0.49) ABL1MAPTRAB9ALMNAMAPK1
SCHEMBL2453455 0.85 TRPA1 (0.49) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL2450859 0.83 TRPA1 (0.48) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL2439686 0.83 TRPA1 (0.53) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL480792 0.83 TRPA1 (0.61) ABL1MAPTNPC1RAB9API4KB
SCHEMBL2450980 0.83 RAB9A (0.47) ABL1MAPTNPC1RAB9ALMNA
SCHEMBL13570204 0.82 TRPA1 (0.47) ABL1MAPTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed