SCHEMBL244373

SCHEMBL244373

c1ccc(C(c2ccccc2)C2CO2)cc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.59
CHRM4 P08173 2/20 0.59
CHRM5 P08912 2/20 0.59
CHRM1 P11229 2/20 0.59
CHRM3 P20309 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245103 1.00 CHRM2 (0.59) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL247653 1.00 CHRM2 (0.59) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17802359 0.88 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17802361 0.88 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17802339 0.88 CHRM1 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17814911 0.88 CHRM2 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL17802337 0.88 CHRM1 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL244385 0.82
SCHEMBL3397822 0.82
SCHEMBL242417 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 91 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016088138-A1 DIPHENYLOXIRANES, PROCESS FOR PREPARATION THEREOF, AND ITS USE IN AN ENANTIOSELECTIVE SYNTHESIS OF (+)-SERTRALINE COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-06-09 WO claimed
US-11453677-B2 Tricyclic compounds useful to treat orthomyxovirus infections NOVARTIS AG (CH) 2022-09-27 US disclosed
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2022-06-30 US disclosed
US-20210186969-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-06-24 US disclosed
EP-3426656-B1 TRICYCLIC COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2021-05-12 EP disclosed
US-10980805-B2 Aza-pyridone compounds and uses thereof Janssen Biopharma, Inc. (US) 2021-04-20 US disclosed
US-10858366-B2 Tricyclic compounds useful to treat orthomyxovirus infections NOVARTIS AG (CH) 2020-12-08 US disclosed
US-20200347072-A1 Tricyclic Compounds Useful to Treat Orthomyxovirus Infections NOVARTIS AG (CH) 2020-11-05 US disclosed
EP-3030566-B1 7,8-DIHYDRO-3H-PYRAZINO[1,2-B]PYRIDAZINE-3,5(6H)-DIONE COMPOUNDS AND USES THEREOF JANSSEN BIOPHARMA INC (US) 2020-07-08 EP disclosed
US-10702523-B2 AZA-pyridone compounds and uses thereof Janssen Biopharma, Inc. (US) 2020-07-07 US disclosed
WO-2002000631-A2 BENZHYDRYL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-03 WO disclosed
EP-1154764-A1 EPOXIDE HYDROLASE COMPLEXES AND METHODS THEREWITH THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2001-11-21 EP disclosed
WO-2000048593-A1 EPOXIDE HYDROLASE COMPLEXES AND METHODS THEREWITH THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-08-24 WO disclosed
EP-0794230-B1 Curable composition based on silyl-functionalized polyethers and epoxy resins KANEKA CORP (JP) 1999-11-10 EP disclosed
US-5889124-A CONSISTS OF AN OXYALKYLENE POLYMER WITH ATLEAST ONE SILICON CONTAINING GROUP HAVING ATLEAST ONE HYDROXYL OR HYDROLYZABLE GROUP BONDED TO A SILICON ATOM, AN EPOXY RESIN, A KETIMINE COMPOUND AND AN ALDEHYDE OR KETONE COMPOUND KANEKA CORPORATION (JP) 1999-03-30 US disclosed
CN-1201919-A Production process of colored fine particulate composition and colored fine particulate composition produced by process DAINICHISEIKA COLOR CHEM (JP) 1998-12-16 CN disclosed
EP-0794230-A2 Curable composition based on silyl-functionalized polyethers and epoxy resins Kaneka Corporation (JP) 1997-09-10 EP disclosed
CN-1107586-A Toner and developer for developing electrostatic image, process for production thereof and image forming method CANON KK (JP) 1995-08-30 CN disclosed
US-4113972-A ANTIDEPRESSANTS BEECHAM GROUP LIMITED (GB) 1978-09-12 US disclosed
US-4101676-A Diphenylpropylamines to treat depression BEECHAM GROUP LIMITED (GB) 1978-07-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10858366-B2 Tricyclic compounds useful to treat orthomyxovirus infections ZC3HAV1, OTC, THOP1 CHRM2 2939/4885CHRM4 2172/4885CHRM5 2630/4885
US-10980805-B2 Aza-pyridone compounds and uses thereof PNPO, ITPA, PDXK CHRM2 359/4885CHRM4 109/4885CHRM5 266/4885
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 CHRM2 508/4885CHRM4 306/4885CHRM5 288/4885
US-20210186969-A1 AZA-PYRIDONE COMPOUNDS AND USES THEREOF PNPO, ITPA, PDXK CHRM2 359/4885CHRM4 109/4885CHRM5 266/4885
US-20200347072-A1 Tricyclic Compounds Useful to Treat Orthomyxovirus Infections ZC3HAV1, OTC, THOP1 CHRM2 2596/4885CHRM4 1810/4885CHRM5 2284/4885
US-10702523-B2 AZA-pyridone compounds and uses thereof PNPO, ITPA, PDXK CHRM2 359/4885CHRM4 109/4885CHRM5 266/4885
US-11453677-B2 Tricyclic compounds useful to treat orthomyxovirus infections ZC3HAV1, OTC, THOP1 CHRM2 2596/4885CHRM4 1810/4885CHRM5 2284/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.