SCHEMBL2446043

SCHEMBL2446043

C[C@@H]1CN(C(=O)O)[C@](c2nc3cc(-c4ccc(Br)cc4)ccc3[nH]2)(C(C)(C)C)C1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.32
HCRTR2 O43614 3/20 0.32
IDO1 P14902 3/20 0.32
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
KIT P10721 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2454367 0.86 GABRA1 (0.31)
SCHEMBL2386864 0.84 PRKCZ (0.31)
SCHEMBL2387383 0.78 GPR119 (0.33)
SCHEMBL2413611 0.78
SCHEMBL1293968 0.77 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL16767137 0.76 CDC7 (0.34)
SCHEMBL2411410 0.74 HRH4 (0.40) IDO1MEN1POLBKMT2A
SCHEMBL1914291 0.74
SCHEMBL1914244 0.74
SCHEMBL2373487 0.72 DAGLA (0.34) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119853-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-29 WO disclosed