SCHEMBL2446255

SCHEMBL2446255

COCCNS(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.75
LMNA P02545 3/20 0.75
HPGD P15428 2/20 0.75
KDM4E B2RXH2 2/20 0.75
NPC1 O15118 1/20 0.75
MAPT P10636 1/20 0.75
RAB9A P51151 1/20 0.75
SMN1; SMN2 Q16637 1/20 0.75
CA12 O43570 6/20 0.67
CA1 P00915 6/20 0.67
CA2 P00918 6/20 0.67
CA9 Q16790 6/20 0.67
HTT P42858 2/20 0.67
ALOX15 P16050 1/20 0.67
CYP3A4 P08684 1/20 0.64
PKM P14618 2/20 0.60
MEN1 O00255 1/20 0.60
POLB P06746 1/20 0.60
TSHR P16473 1/20 0.60
KMT2A Q03164 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20090510 0.91 ALDH1A1 (0.62) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL3699464 0.90 MAPK1 (0.71) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL12302132 0.84 ALDH1A1 (0.90) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL19454404 0.83 ALDH1A1 (0.71) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL19580347 0.83 ALDH1A1 (0.71) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL24762147 0.83 ALDH1A1 (0.75) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL3126117 0.83 ALDH1A1 (0.75) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL386724 0.83 ALDH1A1 (0.75) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL31014207 0.83 ALDH1A1 (0.75) ALDH1A1LMNAHPGDKDM4ENPC1
SCHEMBL29967391 0.83 ALDH1A1 (0.75) ALDH1A1LMNAHPGDKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024243485-A1 CDK2 INHIBITORS AND USES THEREOF ODYSSEY THERAPEUTICS, INC. (US) 2024-11-28 WO disclosed
US-20230062022-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC (US) 2023-03-02 US disclosed
US-11174252-B2 Heterocyclic compounds as kinase inhibitors NUVATION BIO INC. (US) 2021-11-16 US disclosed
CN-112334451-A Heterocyclic compounds as kinase inhibitors 诺维逊生物股份有限公司 2021-02-05 CN disclosed
EP-3752491-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Nuvation Bio Inc. (US) 2020-12-23 EP disclosed
US-10752624-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2020-08-25 US disclosed
WO-2019161224-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS GiraFpharma LLC (US) 2019-08-22 WO disclosed
US-20190248774-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS SAGARD HOLDINGS MANAGER LP, AS ADMINISTRATIVE AGENT (CA) 2019-08-15 US disclosed
US-20180305356-A1 NOVEL KINASE INHIBITORS ORIGENIS GMBH (DE) 2018-10-25 US disclosed
US-10000482-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2018-06-19 US disclosed
US-6855719-B1 Imidazo[1,2-A]pyridine and pyrazolo[2,3-A]pyridine derivatives ASTRAZENECA AB (SE) 2005-02-15 US disclosed
US-20040198757-A1 2-anilino-pyrimidine derivatives as cyclin dependent kinase inhibitors ASTRAZENECA AB (SE) 2004-10-07 US disclosed
US-20040110775-A1 Cyclin dependent kinase inhibiting purine derivatives CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2004-06-10 US disclosed
US-20040106574-A1 2-Arylamino-pyrimidines for the treatment of gsk3-related disorders ASTRAZENECA AB (SE) 2004-06-03 US disclosed
EP-1406876-A1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS Astrazeneca AB (SE) 2004-04-14 EP disclosed
US-20030216406-A1 Pyrimidine derivatives ASTRAZENECA AB (SE) 2003-11-20 US disclosed
EP-1353922-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES Cancer Research Technology Limited (GB) 2003-10-22 EP disclosed
EP-1214318-B1 IMIDAZO[1,2-A]PYRIDINE AND PYRAZOLO[2,3-A]PYRIDINE DERIVATIVES ASTRAZENECA AB (SE) 2003-10-08 EP disclosed
WO-2002096887-A1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS ASTRAZENECA AB (SE) 2002-12-05 WO disclosed
WO-2002059125-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2002-08-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11174252-B2 Heterocyclic compounds as kinase inhibitors CDK6, CDK4, CDK9 ALDH1A1 2534/4885LMNA 2478/4885HPGD 584/4885
US-20040106574-A1 2-Arylamino-pyrimidines for the treatment of gsk3-related disorders GSK3A, GSK3B, CKS2 ALDH1A1 3696/4885LMNA 1157/4885HPGD 2161/4885
US-20180305356-A1 NOVEL KINASE INHIBITORS LRRK2, MYLK2, MYLK ALDH1A1 4333/4885LMNA 3015/4885HPGD 4082/4885
US-20190248774-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS CDK4, CDK6, CDK8 ALDH1A1 2992/4885LMNA 3004/4885HPGD 556/4885
US-20040198757-A1 2-anilino-pyrimidine derivatives as cyclin dependent kinase inhibitors CCNT1, CCNI, CDK2 ALDH1A1 1217/4885LMNA 863/4885HPGD 1342/4885
US-20230062022-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS CDK4, CDK6, CDK8 ALDH1A1 2992/4885LMNA 3004/4885HPGD 556/4885
US-20040110775-A1 Cyclin dependent kinase inhibiting purine derivatives CCNA1, CDKL1, CCNK ALDH1A1 2396/4885LMNA 345/4885HPGD 2212/4885
US-10000482-B2 Kinase inhibitors LRRK2, MYLK2, MYLK ALDH1A1 4184/4885LMNA 3115/4885HPGD 4156/4885
US-20030216406-A1 Pyrimidine derivatives TYMP, TYMS, CCNT1 ALDH1A1 482/4885LMNA 2359/4885HPGD 920/4885
US-10752624-B2 Kinase inhibitors LRRK2, MYLK2, MYLK ALDH1A1 4184/4885LMNA 3115/4885HPGD 4156/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.