SCHEMBL2446469

SCHEMBL2446469

COc1ccc(NC(=O)C2CCCNC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.59
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53
ULK1 O75385 1/20 0.53
POLB P06746 2/20 0.52
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
MAP2K1 Q02750 1/20 0.50
ACHE P22303 1/20 0.50
BACE1 P56817 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2449555 0.85 F10 (0.64) ALOX15NPC1RAB9AULK1POLB
SCHEMBL2448229 0.85 ULK1 (0.56) ALOX15RAB9AULK1
SCHEMBL5205624 0.84 NPC1 (0.69) NPC1RAB9AHPGDHTTPOLB
SCHEMBL23390173 0.83 HTR2C (0.59) ALOX15NPC1HTTULK1POLB
SCHEMBL4564743 0.83 ULK1 (0.64) ALOX15RAB9AHPGDULK1
SCHEMBL8199064 0.83 SMN1; SMN2 (0.64) NPC1RAB9AHPGDHTTPOLB
SCHEMBL3188745 0.83 ENPP3 (0.69) NPC1RAB9AHPGDHTTMTNR1A
SCHEMBL2451482 0.82 ULK1 (0.56) NPC1RAB9AHTTULK1POLB
SCHEMBL2449552 0.82 ULK1 (0.56) ALOX15NPC1RAB9AULK1POLB
SCHEMBL2446479 0.81 HPGD (0.66) ALOX15HPGDULK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed