SCHEMBL5205624

SCHEMBL5205624

COc1ccc(NC(=O)C2CCCC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.69
RAB9A P51151 2/20 0.69
ENPP3 O14638 2/20 0.67
ENPP1 P22413 2/20 0.67
HTT P42858 1/20 0.66
PTPN1 P18031 1/20 0.65
ENPP2 Q13822 1/20 0.63
MTNR1A P48039 1/20 0.63
MTNR1B P49286 1/20 0.63
HPGD P15428 1/20 0.62
STS P08842 1/20 0.62
EPHX1 P07099 1/20 0.61
EPHX2 P34913 1/20 0.61
ACHE P22303 1/20 0.61
BACE1 P56817 1/20 0.61
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
POLB P06746 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3188745 0.98 ENPP3 (0.69) NPC1RAB9AENPP3ENPP1HTT
SCHEMBL8324607 0.93 MTNR1A (0.71) NPC1RAB9AHTTMTNR1AMTNR1B
SCHEMBL18877691 0.90 RAB9A (0.64) NPC1RAB9AENPP3ENPP1HTT
SCHEMBL18877692 0.90 RAB9A (0.64) NPC1RAB9AENPP3ENPP1HTT
SCHEMBL3995294 0.89 ENPP3 (0.59) NPC1RAB9AENPP3ENPP1HTT
SCHEMBL30518933 0.87 MTNR1A (0.64) NPC1RAB9AHTTMTNR1AMTNR1B
SCHEMBL8199064 0.86 SMN1; SMN2 (0.64) NPC1RAB9AHTTMTNR1AMTNR1B
SCHEMBL3197659 0.86 MTNR1A (0.63) NPC1RAB9AHTTMTNR1AMTNR1B
SCHEMBL3197669 0.86 MTNR1A (0.63) NPC1RAB9AHTTMTNR1AMTNR1B
SCHEMBL18951296 0.85 NPC1 (0.60) NPC1RAB9AENPP3ENPP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490043-A4 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO INC (US) 2007-05-30 EP claimed
EP-1490043-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS Merck & Co., Inc. (US) 2004-12-29 EP claimed
WO-2003082190-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-10-09 WO claimed