SCHEMBL24469503

SCHEMBL24469503

O=C1c2c(cccc2[N+](=O)[O-])CN1CC1CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.49
GRM2 Q14416 1/20 0.49
ACHE P22303 2/20 0.43
NR1I2 O75469 1/20 0.43
UGCG Q16739 1/20 0.43
PARP2 Q9UGN5 3/20 0.42
S100A4 P26447 2/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.39
MCL1 Q07820 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
PTPRC P08575 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033749 0.95 PARP1 (0.47) PARP1GRM2ACHENR1I2UGCG
SCHEMBL4024231 0.94 PARP1 (0.46) PARP1GRM2ACHENR1I2UGCG
SCHEMBL4033048 0.92 PARP1 (0.46) PARP1GRM2ACHENR1I2UGCG
SCHEMBL29695767 0.80 ACHE (0.44) PARP1ACHEPARP2S100A4KMT2A
SCHEMBL4029942 0.80 LMNA (0.56) PARP1ACHEPARP2KMT2AMEN1
SCHEMBL14348205 0.78 PARP1 (0.57) PARP1ACHEPARP2KMT2AMAPT
SCHEMBL2333872 0.78 PARP1 (0.48) PARP1ACHES100A4KMT2AMAPT
SCHEMBL4209630 0.78 ACHE (0.43) PARP1ACHEPARP2S100A4KMT2A
SCHEMBL4026308 0.77 PARP1 (0.48) PARP1ACHEPARP2KMT2AMEN1
SCHEMBL24469636 0.77 PARP1 (0.56) PARP1NR1I2UGCGPARP2CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115301-A1 MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2022-06-02 WO disclosed