SCHEMBL14348205

SCHEMBL14348205

O=C1c2c(cccc2[N+](=O)[O-])CN1Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.57
PREP P48147 7/20 0.53
ACHE P22303 2/20 0.46
POLB P06746 1/20 0.44
PARP2 Q9UGN5 1/20 0.43
MAPT P10636 2/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
MCL1 Q07820 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ATM Q13315 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2333872 0.92 PARP1 (0.48) PARP1PREPACHEMAPTRECQL
SCHEMBL3910578 0.86 PARP1 (0.44) PARP1PREPACHEMAPTRECQL
SCHEMBL31281346 0.85 DCTPP1 (0.48) PARP1PREPKMT2A
SCHEMBL4029942 0.80 LMNA (0.56) PARP1ACHEPOLBPARP2MAPT
SCHEMBL29695767 0.80 ACHE (0.44) PARP1ACHEPARP2MAPTRECQL
SCHEMBL2024995 0.79 PARP1 (0.64) PARP1PREPPARP2
SCHEMBL24469503 0.78 PARP1 (0.49) PARP1ACHEPARP2MAPTRECQL
SCHEMBL4209630 0.78 ACHE (0.43) PARP1ACHEPOLBPARP2MAPT
SCHEMBL14348206 0.78 DHPS (0.54) ACHEPOLBMAPTRECQLKMT2A
SCHEMBL2030975 0.78 KMT2A (0.43) ACHEPOLBMAPTRECQLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312214-B2 1, 1-disubstituted cycloalkyl derivatives as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-12-25 US disclosed