SCHEMBL24503136

SCHEMBL24503136

O=C(c1ccc(F)cc1)N1Cc2ccc(Br)cc2C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRAP1 Q12931 3/20 0.53
HSP90B1 P14625 2/20 0.53
HSD11B1 P28845 2/20 0.51
ABHD6 Q9BV23 1/20 0.50
NAMPT P43490 4/20 0.46
HPGD P15428 1/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
DPP8 Q6V1X1 1/20 0.45
DPP9 Q86TI2 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
GPR183 P32249 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
KMT2A Q03164 1/20 0.45
DRD1 P21728 1/20 0.44
PTGER2 P43116 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
KLKB1 P03952 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24503025 0.89 ABHD6 (0.54) HSD11B1ABHD6NAMPTHPGDLMNA
SCHEMBL4505014 0.86 ABHD6 (0.48) TRAP1HSP90B1ABHD6NAMPTHPGD
SCHEMBL26525246 0.81 GPR183 (0.51) ABHD6NAMPTHPGDDPP8DPP9
SCHEMBL24685025 0.77 TRAP1 (0.55) TRAP1HSP90B1NAMPTHPGDDPP8
SCHEMBL4437450 0.75 ABHD6 (0.55) ABHD6NAMPTDPP8DPP9DPP7
SCHEMBL1956852 0.75 ABHD6 (0.55) ABHD6NAMPTDPP8DPP9DPP7
SCHEMBL18085956 0.74 TRAP1 (0.55) TRAP1HSP90B1NAMPTKDM4EMEN1
SCHEMBL16101941 0.74 NOTUM (0.60) ABHD6NAMPTDPP8DPP9DPP7
SCHEMBL20439780 0.74 HPGD (0.59) ABHD6NAMPTHPGDLMNAHTT
SCHEMBL25592808 0.73 CA12 (0.44) TRAP1HSP90B1HSD11B1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4257588-A1 SMALL MOLECULE INHIBITOR OF CATHEPSIN C AND MEDICINAL USE THEREOF Reistone Biopharma Company Limited (CN) 2023-10-11 EP disclosed
WO-2022117059-A1 SMALL MOLECULE INHIBITOR OF CATHEPSIN C AND MEDICINAL USE THEREOF 瑞石生物医药有限公司 2022-06-09 WO disclosed