SCHEMBL24508992

SCHEMBL24508992

O=CNc1ccc2c(c1)OCC(=O)N2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.54
TRPV1 Q8NER1 1/20 0.50
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
IDH1 O75874 1/20 0.46
MMP12 P39900 1/20 0.45
PKM P14618 3/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA5 P31644 1/20 0.45
CYP3A4 P08684 2/20 0.45
CYP19A1 P11511 2/20 0.45
CYP2C9 P11712 2/20 0.45
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PARP1 P09874 3/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28105822 0.88 ALDH1A1 (0.59) TRPV1ALDH1A1MAPTMMP12PKM
SCHEMBL12362001 0.81 KIF11 (0.56) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL23432581 0.79 KIF11 (0.54) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL3027487 0.78 CYP11B1 (0.50) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL6297431 0.77 KIF11 (0.62) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL3594625 0.76 MMP12 (0.51) KIF11ALDH1A1MAPTCYP11B1CYP11B2
SCHEMBL4578101 0.75 TRPV1 (0.56) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL10269414 0.75 KIF11 (0.60) KIF11TRPV1CYP11B1CYP11B2IDH1
SCHEMBL17315403 0.75 KIF11 (0.54) KIF11TRPV1ALDH1A1MAPTCYP11B1
SCHEMBL9033589 0.75 PARP1 (0.55) KIF11MAPTCYP11B1CYP11B2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022123039-A1 ALDEHYDE DEHYDROGENASE INHIBITORS AND THEIR THERAPEUTIC USE CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-06-16 WO disclosed