SCHEMBL2451499

SCHEMBL2451499

Cn1c(=O)n(C)c2nccn2c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
PDE4A P27815 4/20 0.33
PDE4B Q07343 4/20 0.33
PDE4C Q08493 4/20 0.33
PDE4D Q08499 4/20 0.33
PDE1A P54750 2/20 0.33
PDE1B Q01064 2/20 0.33
PDE1C Q14123 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PIK3CD O00329 2/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA2B P29275 2/20 0.32
ADORA1 P30542 2/20 0.32
POLB P06746 1/20 0.32
CNR1 P21554 1/20 0.32
ACHE P22303 1/20 0.32
NTSR1 P30989 1/20 0.32
MC3R P41968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22071869 0.65 ADORA3 (0.36) CCNE1CDK2PDE4APDE4BPDE4C
SCHEMBL12799838 0.65 DDB1 (0.41) ADORA2BADORA1ALDH1A1
SCHEMBL8345010 0.63 ALDH1A1 (0.35) PDE4DPDE1APDE1BPDE1CHSD17B10
SCHEMBL8345008 0.63 AAK1 (0.35) HPGDALDH1A1MAPT
SCHEMBL20780218 0.63
SCHEMBL13936549 0.62 ADORA3 (0.41) CCNE1CDK2PDE4APDE4BPDE4C
SCHEMBL7481984 0.61 PDE4A (0.36) CCNE1CDK2PDE4APDE4BPDE4C
SCHEMBL21912931 0.61
SCHEMBL22071854 0.58 ADORA3 (0.33) ADORA3
SCHEMBL22072415 0.58 ADORA3 (0.33) ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed